Zaj tshaj tawm
Cov tshuaj no tau txwv tsis pub muag, peb lub vev xaib tsuas tuaj yeem tshawb xyuas cov ntaub ntawv yooj yim. Tshuaj ntawm no, peb tsis muag lawv!
Lub Kaum Hli 22, 2024
Anavar Hmoov, tseem hu ua Oxandrolone, Dawb tsis muaj ntxhiab crystalline hmoov, soluble hauv ethanol, acetone, me ntsis soluble nyob rau hauv ether, soluble me ntsis hauv dej. Analar yog lub suab hluavtaws meloic steroid. Cov qauv molecular yog c13h16d2o2, nrog lub cev hnyav molecular ntawm 216.31. Cov pa roj carbon (c) nyiaj rau 47.48%, Hydrogen (H) Accounts rau 5.48%, deuterium (d) account rau 3.06%, thiab cov pa) rau 29.06%. Nws yog ib tus dawb rau ze li dawb crystalline hmoov. Tsis txhob yaj ntawm chav sov, nrog lub ntsiab lus melting ntawm kwv yees li 253 degree C. nkag siab txog lub teeb, kub, thiab huab cua, ntev ua rau huab cua tuaj yeem ua rau cov xim hloov xim. Nws tuaj yeem raug siv los ua assimation tus neeg sawv cev hauv Biomedical kev tshawb fawb los txhawb cov protein synthesis thiab kev loj hlob ntawm tes. Nws tseem siv los kawm cov kev cuam tshuam ntawm cov tshuaj hormones ntawm kev loj hlob ntawm tes thiab kev sib txawv, nrog rau kev tshawb nrhiav kev kho mob rau cov kabmob muaj feem xyuam. Nws tseem muaj qee daim ntawv thov tus nqi hauv kev tshawb fawb tshuaj thiab kev loj hlob. Piv txwv li, nws tuaj yeem siv los kawm cov txiaj ntsig ntawm cov tshuaj ntawm cov leeg kev loj hlob thiab rov zoo, lossis ua tus qauv rau kev tsim tshuaj thiab kev ua kom zoo. Nws tuaj yeem raug siv ua tus qauv sab hauv lossis cov qauv hauv kev kuaj mob tshuaj ntsuam xyuas kom ntsuas kev pom zoo thiab faib lwm cov sib txuas ua ke hauv cov qauv biochemical.
Phem (oxandrolone) yog cov tshuaj shau tshuaj steroid uas tuaj yeem siv los kho ntau yam kab mob thiab cov tsos mob.
Cov hauv qab no yog cov tshuaj tseem ceeb ntawm Anavar:
(1) Kev Kho Mob Atroph Cov tsos mob: Anavar tuaj yeem txhawb cov leeg kev loj hlob thiab nce cov leeg kom muaj zog thiab qhov zoo. Yog li ntawd, nws feem ntau yog siv los kho cov leeg mob atrophy itty tshwm sim los ntawm ntau yam, xws li kub hnyiab, kev raug mob, kev phais mob, kev phais, thiab lwm yam.
(2) Kev Kho Mob Osteoporosis: Anavar tuaj yeem nce pob txha ceev thiab pob txha morphology, yog li txo qhov kev pheej hmoo ntawm cov mob easteoporosis.
(3) Nce cov ntshav liab liab suav: Anavar tuaj yeem tsim kev ntau lawm cov ntshav liab, yog li ua kom cov tsos mob ntshav ntshav liab.
(4) txo cov rog lub cev: Aavar tuaj yeem txhim kho cov metabolic tus nqi, txo cov kev sib txuam ntawm cov rog hauv lub cev, thiab txhim kho cov rog rog.
Nyob rau ntawm Anavar muag online, peb cov kws tshawb nrhiav hauv chav kuaj siv tshuaj lom neeg tshuab oxandrolone synthesis. Koj tuaj yeem so kom paub tseeb tias anavar siv.
Tshuaj Cov Qauv |
C19H30O3 |
Muaj pes tsawg leej |
306 |
Molecular hnyav |
306 |
m/z |
306 (100.0%), 307 (20.5%), 308 (2.0%) |
Kev Ntsuam Xyuas |
C, 46.81; H, 6.07; Cl, 25.12; N, 4.96; O, 5.67; S, 11.36 |
Morphological |
hmoov |
Xim |
dawb rau beige |
Melting taw tes |
235-238 degree c |
Kub taw tes |
387.04 DEGREES (Kwv TAIS |
Ceev |
1.0829 (ntxhib kwv yees) |
Kev Cia |
2-8 degree c |
Solubility Cawv |
40 ntu ntawm cov kuab tshuaj |
Acidity Coefficient (PKA) |
15.15 {{{0. 60 (kwv yees) |
Solubility H2o |
2mg / ml (kev daws teeb meem; ua kom sov) |
Kev ua kho qhov muag [] |
D -19 rau -26 degree, c=1 (cdcl3) |
Refronction Index |
1.4200 (kwv yees) |
Peb tuaj yeem muab khoomAnavar Hmoov.
Cov lus hais: Bloom Tech (Txij xyoo 2008), ua tiav chem-tech yog tus muab kev pabcuam ntawm peb.
Anavar yog qhov ncauj lus hluavtaws siv los txhim kho cov leeg loj hlob thiab txhawb kev txhim kho pob txha.
Cov hauv qab no yog qhov muaj peev xwm anavar synthesis txoj kev:
(1) Ua ntej, Acetophenone yog siv nrog acetic anhydride kom tsim Ester.
(2) oxidize tus ester nrog molecule ntawm acetic acid, ib qho molecule ntawm cov dej {}} mehle}} mehle}}} CIS-enone.
(3) {2- hydroxy {2}}}}}}}}}}}}} {} Methyl {12}} xohydroispoisoxazole.
(5) Ntxiv 5 -}}}} methyl {}} hydroxide yog rhuab los ua anavar.
Methylprednisolone tau nrawm nrawm los ntawm kev tswj hwm plab zom mov. Nws cov metabolites thiab cov pa roj oxygen thiab cov pa roj carbon monoxusgen ib txwm tau ua los ntawm Shen thiab ib tus nqi me me yog ua rau txoj hnyuv. Kev loj hlob thiab kev kawm tiav nyob rau hauv cov tub thiab Orgenital Ovarian hypoplasia hauv cov ntxhais (tshuaj ntsuam mob) * Cov thawj coj tuaj yeem ua rau pom tseeb. Cov uas muaj lub siab ua hauj lwm yuav tsum tsis txhob siv oxymethylprednisolone.
Keeb kwm txhim kho ntawmAnavar Hmoov:
(1) Hauv xyoo 1964, Anavar tau ua ke los ntawm cov nom tswv chaw ua hauj lwm (tam sim no ib ceg ntawm Pfizer). Thaum pib, nws tau siv los kho cov mob epeeoporosis thiab cov leeg leeg atrophy, hlawv, postoperative rov qab, thiab lwm yam.
(2) Anavar yog nrov heev vim tias nws muaj qis qis toxicity thiab tsawg dua kev phiv puas dua li lwm cov tshuaj steroids. Txawm li cas los xij, nyob rau xyoo 1980 thiab 1990s, kev tsim khoom thiab muag ntawm Anavar tau raug tshem tawm vim kev tsim txom, muag khoom tsis raug cai thiab kev raug teeb meem raug rho tawm.
(3) Hauv xyoo 1995, lub tuam txhab uas tsim thiab muag Anavar pib tsim ib lub cev ib yam ntxiv. Tam sim no, Anavar yog siv los kho ntau cov leeg mob atrophy aimphy, xws li tus kabmob HIV, tshuaj khomob, thiab lwm yam.
Tsis tas li ntawd, vim tias nws tuaj yeem nce cov leeg loj hlob, ua kom lub cev muaj zog, ua kom cov neeg ncaws pob, tab sis nws txoj kev raug mob thiab tsis raug cai ua rau muaj kev pheej hmoo txaus ntshai. Thov nco ntsoov tias cov khoom no yog rau kev kuaj siv nkaus xwb.
Anavar Hmoovyog cov hluavtaws metabolic steroid nrog ntau yam molecular tus yam ntxwv. Hauv qab no yog cov yam ntxwv tseem ceeb ntawm Anavar cov qauv txheej txheem:
1. {{{{{}} And}}}}}}}}} methyl thiab {{9 {9}} cawv {{} ketone thiab lwm yam qauv txheej txheem. Qhov kev npaj cov kev cai tshwj xeeb no tso nws nrog kev siv hluav taws xob metabolic. 2. Cov pa oxygen atomes roj carbon ib hauv dihydrotestosterone: piv rau DHT molecule los ntawm kev ntxiv cov pa otom rau ob cov roj av atom. Cov kev qhia txog cov pa oxygen no txhim kho nws cov nyhuv anabolic, ua rau muaj kev ntsuas siab dua li DHT.
3. Methyl Group Hloov 17 carbon atoms: 17 roj teeb atoms: 17 carbon atoms hauv Anavar lwg me me tau hloov los ntawm cov pab pawg methyl. Kev hloov methylation no ua rau Anavar C17 Anabolic Steroid, raws li feem ntau c17 Anabolic cov tshuaj steroids nyuaj rau nqus tau qhov ncauj lus.
4. Attinity nrog Androgen cov qauv: Anavar cov qauv molecular muaj kev sib txuas lus siab, yog li txhawb nqa cov kab mob transductioncution
5. Txo metabolic kev ua si: Vim qee qhov kev hloov pauv ntawm Anaval Molecule, yog li txo qhov tau ntawm nws cov kev sib tsoo metabolic hauv lub cev. Qhov no pab txuas ntxiv lub sijhawm ntawm nws cov txiaj ntsig thiab txo qhov ntau zaus ntawm kev siv.
Dab tsi yog cov kev phiv los ntawm no compound no?
1.Liver Toxicity
Anavar yog c -17} epha alkylated steroid, thiab nws tus qauv muab nws hepatotoxicity. Txawm hais tias Anavar muaj qis dua daim siab ua kom mob siab sib piv rau lwm tus, ntev ntev yuav ua rau lub siab puas.
Lub siab ua kom lub siab enzymes
Tom qab siv Anavar, cov neeg mob tuaj yeem muaj kev nce siab nyob hauv daim siab enzymes xws li ist thiab alt, uas feem ntau qhia qee qhov kev sim siab.
Cov qib ntawm lub siab Enzymes sib txawv ntawm cov tib neeg, tab sis feem ntau maj mam rov qab thaum siv Anavar lossis tom qab ua kom tsis zoo.
Yog tias lub siab ua kom lub siab tsis tu ncua lossis paug, nws yuav tsim nyog kom tsis txhob siv Anavar thiab yauv mus tom qab daim siab kuaj ntshav.
Mob siab Kab Mob
Tsawg tsawg zaus, siv sijhawm ntev ntawm Anavar yuav ua rau muaj kab mob siab xws li cov kab mob cirrhosis lossis purpura muaj kab mob siab.
Cov kab mob no tuaj yeem ua rau lub siab tsis ua tiav thiab txawm tias muaj kev phom sij lub neej.
Yog li ntawd, thaum siv Anavar, cov neeg mob yuav tsum tau saib xyuas lub siab thiab saib xyuas ib qho kev mob siab, xws li mob taub hau, mob plab, thiab lwm yam.
2.Txhob rau ntawm cov hlab plawv
Anavar yuav muaj qee qhov teebmeem ntawm cov hlab plawv, suav nrog kev hloov pauv ntshav siab thiab cov qib roj cholesterol.
Txhawb cov ntshav siab
Anavar yuav ua rau cov ntshav nce siab, uas tej zaum yuav yog vim nws cov nyhuv ntawm kev ua kom cov qe ntshav liab ntau thiab ntshav viscosity.
Tawg siab yuav ua rau muaj kev pheej hmoo mob plawv thiab mob stroke.
Cov neeg mob uas muaj keeb kwm kev kub siab yuav tsum ceev faj thaum siv Anavar thiab saib xyuas lawv cov ntshav siab.
Hloov pauv cov roj (cholesterol)
Anavar yuav ua rau muaj kev nce lipoprotein tsawg (LDL,
Qhov kev hloov no hauv cov qib roj cholesterol yuav ua rau muaj kev pheej hmoo ntawm atherosclerosis, uas nyeg ua rau muaj kev pheej hmoo mob plawv.
Yog li ntawd, thaum siv Anavar, cov neeg mob yuav tsum tau cov ntshav ntsuas lipid tsis tu ncua thiab / lossis siv tshuaj lipid-txo raws li tus kws kho mob cov lus qhia.
3. Tu neeg kaw lus kaw lus
Anavar, raws li ib daim ntawv ntawm exogenous Testosterone, tej zaum yuav muaj qee yam cuam tshuam ntawm cov txheej txheem endocrine, suav nrog ua rau muaj kev sib deev endogenous testosterone ntau lawm thiab hloov deev cov xim deev endogenous thiab hloov deev hom somon.
Inhibition ntawm endogenous Testosterone Ntau Lawm
Anavar yuav inhibit txoj haujlwm ntawm hypothalic temuitary gonadal gonadal axis, yog li txo endogenous Testosterone ntau lawm.
Qhov kev cuam tshuam no yuav ua rau cov tsos mob sib deev xws li tsawg dua Libido thiab erectile kawg.
Siv sijhawm ntev ntawm Anavar yuav ua rau muaj kev sim siab thiab txo cov phev suav.
Hloov pauv ntawm cov qib kev sib deev Hormone
Anavar yuav nce cov qib tshuaj estrogen (txawm hais tias nws cov nyhuv muaj zog tsis muaj zog), uas yuav ua rau cov tsos mob xws li txiv neej lub mis loj (feminization) thiab Edema.
Nyob rau tib lub sijhawm, Anavar kuj tseem tuaj yeem nce cov progesterone (xws li progesterone), uas yuav ua rau qee lub suab thiab cov plaub hau qis (txawm hais tias tsis tshua muaj poj niam).
4.Skin teeb meem
Anavar yuav muaj qee yam teebmeem ntawm daim tawv nqaij, suav nrog pob txuv, plaub hau, thiab lwm yam.
Pob kab ntxaus
Anavar yuav nce daim tawv nqaij tso pa tawm, ua pob txuv.
Acne feem ntau tshwm nyob rau hauv cov chaw muaj ntau cov qog sebaceous xws li lub ntsej muag, rov qab, thiab lub hauv siab.
Rau cov neeg mob uas twb muaj pob txuv, siv Anavar yuav ua rau cov tsos mob tshwm sim.
Alopecia
Anavar yuav ua rau nce qib DHT (Dihydrotestosterone), ib qho tshuaj hormones uas ua rau txiv neej hom plaub hau poob.
Siv sijhawm ntev ntawm Anavar yuav ua rau cov tsos mob xws li kev sib kis plaub hau thiab cov plaub hau poob.
Hom plaub hau no feem ntau yog cov khoom siv tshuaj ntsuab, yog li rau cov neeg mob keeb kwm ntawm cov plaub hau poob, siv anavar yuav ua rau muaj kev pheej hmoo ntawm cov plaub hau plaub hau.
Kev cai tswjfwm kev cai lij choj ib puag ncig
Vim tias cov teeb meem kev noj qab haus huv uas cuam tshuam nrog hluavtaws medoolic steroids, ntau lub teb chaws tau siv nruj cov cai kev cai lij choj ntawm cov tshuaj no. Yog li ntawd, kev tsim txoj cai lij choj, muag, thiab siv Anavar yuav raug txwv nruj me ntsis los ntawm cov cai lij choj no thiab cov cai. Nyob rau hauv cov ntsiab lus ntawm stricter kev cai, Anavar cov chaw ua lag luam yuav raug compressed.
Hloov hauv kev ua lag luam xav tau
Txawm hais tias Anavar yuav muaj qee qhov kev xav tau tshwj xeeb hauv qee cov haujlwm tshwj xeeb, kev ua kis las, kev ua kis las, thiab lwm yam thiab hloov kom haum. Piv txwv li, kev nce qib kev paub txog kev noj qab haus huv thiab kev tawm dag zog yuav txhawb nqa lawv lub cev nqaij daim tawv, tsis yog kev vam meej ntawm cov khoom siv metabolic me me. Tsis tas li ntawd, nrog kev nce qib nruam kev siv thev naus laus zis thiab kev txhim kho cov tshuaj tshiab, yuav muaj kev nyab xeeb dua, uas yuav cuam tshuam ntxiv rau kev lag luam xav tau ib lub anavar.
Kev tshawb fawb tshawb fawb thiab kev nce qib thev naus laus zis
Hauv kev tshawb fawb ntawm kev tshawb fawb thiab thev naus laus zis, kev tshawb fawb ntawm cov khoom siv metabolic medoolic thiab cov khoom siv cuam tshuam hluav taws xob thiab cov tshuaj ntsig yuav txuas ntxiv. Cov kev tshawb fawb no yuav qhia tau ntau yam peev xwm siv tau lossis cov kev mob tshwm sim ntawm Anavar, yog li cuam tshuam nws txoj kev txhim kho. Lub caij no, nrog kev nce qib txuas ntxiv ntawm biotechnology thiab tshuaj siv tshuaj, ntau dua cov tshuaj tshiab, uas yuav hloov pauv anavar hauv qee yam.
Cov pej xeem kev xav thiab kev coj ncaj ncees
Ntxiv rau kev cai lij choj thiab kev xav tau lag luam, kev xav txog pej xeem kuj tseem muaj feem cuam tshuam txog kev txhim kho kev cia siab ntawm Anavar. Tawm tsam lub nraub qaum ntawm kev ua kom muaj kev txhawj xeeb txog kev quav tshuaj thiab kev pheej hmoo muaj kev noj qab haus huv, kev siv Anavar yuav ntsib cov lus nug ntxiv thiab kev thuam. Lub siab ntawm cov pej xeem cov pej xeem lub tswv yim yuav muaj qhov cuam tshuam tsis zoo rau nws cov kev lag luam hauv khw.
Cim npe nrov: Anavar Hmoov Li {{53-39-4, cov chaw muag khoom, chaw tsim khoom, Hoobkas, lag luam, yuav khoom, rau muag