Txawm hais tias kev noj haus yog ib qho ntawm cov hloov pauv uas yuav cuam tshuam rau kev ua tau zoo ntawm cov kev ua si flasaner thaum nws los tiv thaiv mub thiab zuam hauv cov dev. Rau qhov zoo tshaj plaws cov txiaj ntsig tau, nws yog qhov tseem ceeb rau cov tswv tsiaj thiab cov kws kho tsiaj kom paub tias kev noj haus yuav cuam tshuam dab tsi cuam tshuam rau kev nqus ntawmNtsesaner ntsiav tshuajCov. Txhawm rau pab koj kom tau tshaj tawm ntawm cov kab mob tshiab no, cov lus qhia ntxaws ntxaws no yuav dhau mus rau txhua txoj hauv kev uas koj tau cuam tshuam ntau npaum li cas fluralaner koj nqus tau ntau npaum li cas.

1.Txoj kev tshwj xeeb (hauv Tshuag)
(1) daws
(2) Ntsiav tshuaj
(3) kev txhaj tshuaj
(4) txau
(5) poob
2.Customization:
Peb yuav sib tham ntawm tus kheej, OEM / ODM, tsis muaj hom, rau kev tshawb nrhiav kev ua haujlwm nkaus xwb.
Code sab hauv: Bm-2-079
Fluralaner CASE 864731-61-3
Kev Lag Luam Tseem Ceeb: Tebchaws Asmeskas, Australia, Nyij Pooj, Tebchaws Yelemees, Indonesia, UK, New Zealand, Canada thiab lwm yam.
Chaw tsim tshuaj paus: BOUAB TECH XI'AN HOOBKAS
Kev tsom xam: HPLC, LC - ms, hnmr
Kev Txhawb Nqa Tshuab: R & Dept.-4
Peb muab cov fluralaner, thov saib mus rau lub vev xaib hauv qab no rau cov ncauj lus qhia ntxaws ntxaws thiab cov ntaub ntawv khoom siv.
Khoom:https://www.bloomteechz.com/Oemixat{2 }oodm/tablet/Fridalaner{erIerIer{herixeMlet.html
Lub Nruab Nrab ntawm kev cuam tshuam ntawm cov khoom noj khoom haus ntawm kev nqus ntawm cov ntsiav tshuaj nplua miasaner
Qhov nqus ntawm cov ntsiav tshuaj fluralaner tuaj yeem cuam tshuam los ntawm lub xub ntiag ntawm cov zaub mov hauv txoj hnyuv plab. Qhov kev sib cuam tshuam no feem ntau vim yog lub pob physicochemical ntawm Fluralaner thiab nws kev sib cuam tshuam nrog ntau yam khoom noj khoom noj. Cia relve rau hauv cov txheej txheem tshwj xeeb uas cuam tshuam cov txheej txheem no:

Lipid - Raws li kev tso siab
Fluralaner yog lipophilic sib xyaw, txhais tau tias nws muaj kev sib raug zoo rau cov rog. Thaum muab cov neeg ua haujlwm siab rau lub siab- cov mov noj muaj roj, qhov nqus ntawm Fluralaner tuaj yeem txhim kho. Qhov no yog vim cov zaub mov muaj rog los txhawb kev tsim cov kua dej bile, uas tuaj yeem siv tshuaj lipophilic zoo li fluralaner thoob plaws plab hnyuv.
Pais plab nchuav cov nqi hloov kho
Lub xub ntiag ntawm cov zaub mov hauv plab tuaj yeem qeeb zuj zus patric khoob, uas nyeg cuam tshuam rau tus nqi ntawm uas fluralaner nce mus rau txoj hnyuv me me. Qhov no qeeb plab nchuav tuaj yeem ua rau muaj kev sib tw ntev dua mus rau qhov chaw nqus, muaj peev xwm nce nws cov bioavailability.
Ph - Yeem Sawv Daws Hloov Hloov
Cov zaub mov noj tuaj yeem hloov cov pH ntawm cov kab mob plab, uas tuaj yeem cuam tshuam rau solubility ntawm fluralaner. Cov tshuaj solubility yog ph - Nyob ntawm, thiab cov kev hloov pauv hauv PH tuaj yeem cuam tshuam nws cov kev sib cais thiab kev nqus tau.
Kev sib piv ntawm Fluralaner Bioavailability nyob rau hauv high - pat} Cov Khoom Noj Rog Rog Vs. Fasted State
Nkag siab txog qhov sib txawv ntawm Fluralaner Bioavailability ntawm kev pub thiab cov xeev yoo mov yog qhov ua kom zoo dua kev kho mob. Ntau cov kev tshawb fawb tau tshawb xyuas qhov no nam, muab cov kev pom zoo nyob rau hauv cov zaub mov muaj kev nqus cov ntsiav tshuaj nqus.
Bioavailability ua kom haum nrog siab - cov zaub mov muaj roj
Kev tshawb fawb tau ua ntu zus uas tswj cov ntsiav tshuaj foodaner nrog lub siab {}} rog tau noj mov ntau dua nws cov txiaj ntsig. Hauv ib qho kev kawm piv, thaj chaw hauv qab nkhaus (AUC) thiab siab tshaj plaws Plasma thiab siab tshaj plaws Plasmaner tau pom tias muaj txiaj ntsig zoo dua thaum muab cov zaub mov muab piv rau lub xeev fasted.

Fasted Lub Xeev Nqus Cov Cwj Pwm
Nyob rau hauv lub xeev fasted, Floraneaner qhov nqus tau feem ntau qis dua thiab ntau dua cov. Qhov no feem ntau yog vim tsis muaj cov zaub mov -}}}}} Qhov kev nqus tshuaj no, xws li kev tso pa tawm hauv cov plab zom mov thiab nce qib siab.
Kev kho mob cuam tshuam ntawm cov zaub mov -} induced Bioavailability hloov
Lub txhim kho cov xyoob ntoo ntawm fluralaner thaum muab cov zaub mov muaj cov khoom noj cuam tshuam tseem ceeb. Nws qhia tias pub cov tsiaj ua ntej lossis thaum lub sijhawm kev kho mob yuav ua rau muaj txiaj ntsig zoo thiab muaj peev xwm ntev dua-} kav tiv thaiv mub thiab zuam. Txawm li cas los xij, nws yog ib qho tseem ceeb kom nco ntsoov tias tusNtsiav tshuaj chew cov xov toojtseem tshuav tib yam tsis hais txog kev tswj hwm cov xwm txheej, ua tus nqi -}}} Xaiv cov tswv tsiaj.
Chaw ua zaub mov ntawm cov chaw noj zaub mov ntawm cov khoom noj ntawm cov khaub thuas ntawm cov ntsiav tshuaj nqus
Lub chaw muag tshuaj ntawm cov fluralaner yog ho cuam tshuam los ntawm cov zaub mov noj, uas tuaj yeem tiv thaiv rau ntau qhov tseem ceeb:
Muaj kev nqus cov cheeb tsam nqus dej
Khoom noj khoom haus thiab kev tso kua dej tso kua roj zom, uas nyeg ua rau lub plab zom mov. Qhov kev ua tau zoo no nthuav dav thaj chaw nqus dej nyob hauv cov hnyuv, uas pub rau kev sib cuam tshuam zoo dua ntawm cov tshuaj, xws li fluralaner, thiab txoj hnyuv plab. Nrog rau thaj chaw loj dua rau kev nqus, cov tshuaj muaj ntau txoj hauv kev los nqus rau hauv cov hlab ntshav, txhim kho nws tag nrho cov bioavailability. Qhov kev sib cuag tau ntau dua ntawm cov tshuaj thiab cov mucosal ob sab phlu yog qhov tseem ceeb rau kev nqus tau zoo, tshwj xeeb tshaj yog rau cov tshuaj uas yuav tsum muaj kev sib cuam tshuam ntau nrog cov hnyuv hnyuv.
Lymphatic kev thauj mus los
Siv cov zaub mov siab high - Cov zaub mov muaj roj tuaj yeem pab txhawb cov lipophilic tshuaj zoo li fluralaner. Tsis zoo li dej - cov tshuaj yeeb tshuaj, cov tshuaj lipophilic yog nqus tau los ntawm lub siab thawj- dhau metabolism. Txoj kev nqus tau txoj hauv kev no tuaj yeem ua rau cov tshuaj ntau dua ntawm cov tshuaj hauv kev ncig ua si, nce nws cov peev xwm. Txoj kev Lymphatics muab txoj hauv kev ncaj qha rau cov tshuaj kom nkag mus rau cov ntshav, tshwj xeeb tshaj yog thaum coj nrog cov khoom noj muaj roj.
Lub Sij Hawm Roj Hnyav Rov Qab Los
Thaum cov zaub mov noj, nws ua rau qeeb qeeb ntawm cov roj hauv plab zom mov, tso cai rau cov tshuaj uas yuav nyob hauv lub plab zom mov rau lub sijhawm ntev dua. Qhov no txuas ntxiv lub sijhawm txhais tau tias Floraner muaj ntau lub sijhawm los cuam tshuam nrog cov chaw nqus dej hauv cov hnyuv, nce nws txoj kev tau nqus mus rau hauv cov hlab ntshav. Kev raug mob dua los ua kom haum cov chaw muaj peev xwm ua rau muaj kev sib tw ntau dua, raws li cov tshuaj muaj ntau txoj hauv kev los ntawm cov hlab ntshav ua ntej kev tshem tawm ntawm lub plab zom mov. Qhov kev pom zoo no tuaj yeem txhim kho cov nyhuv kho mob ntawm cov tshuaj.
Kev tshawb fawb tshawb fawb rau Fluralaner ntsiav tshuaj tswj hwm sijhawm hauv kev siv kho mob
Raws li cov ntaub ntawv tshawb fawb thiab cov kev tshawb nrhiav chaw soj ntsuam, ntau cov lus pom zoo tuaj yeem ua kom txog lub sijhawm zoo ntawmNtsiav tshuaj FluralanerTswjhwm:
FORRYISTERING RAU COV ME NYOOG
Txhawm rau kom ua kom haum thiab ua tau zoo, nws feem ntau pom zoo los tswj cov ntsiav tshuaj Foodaner nrog lossis tam sim ntawd ib qho uas muaj ib txwm muaj cov rog.
Sib xws hauv kev tswj hwm
Rau ntev - Term kev tiv thaiv, tswj kev tiv thaiv kev noj haus thaum lub sijhawm tswj hwm tau ntau cov tshuaj ntau thiab kev ua tau zoo.
Kev txiav txim siab ntawm cov neeg muaj tsiaj
Thaum kev pub mis muaj txiaj ntsig zoo rau kev nqus cov khaub ncaws fluralaner thiab cov khoom noj kom zoo li kev noj qab haus huv thaum txiav txim siab ua haujlwm zoo.
Qhov tseem ceeb ntawm cov khoom noj khoom haus hauv Fluralaner ntsiav tshuaj ntsiav tshuaj
To taub cov khoom noj muaj txiaj ntsig zoo ntawm Fluralaner qhov tseem ceeb rau kev tsim cov lus qhia txog kev txhim kho kev zoo thiab ua kom tau zoo tshaj kho cov txiaj ntsig zoo:
Dose Haum Kev Txiav Txim Siab
Lub zog hloov pauv ntawm fluralaner thaum muab cov khoom noj yuav muaj feem tau noj kev hloov kho hauv qee qhov scorathical. Txawm li cas los xij, nws yog ib qho tseem ceeb kom nco ntsoov tias cov lus pom zoo tam sim no yog nce raws kev kho kom muaj kev nyab xeeb thiab kev hloov kho tau zoo, thiab txhua yam kev hloov kho yuav tsum tau ua raws li kev coj kho tsiaj.
Tus Neeg Mob Kev Kawm
Qhia cov tsiaj tsiaj txog kev cuam tshuam ntawm cov zaub mov ntawm Floraner nqus tuaj yeem txhim kho kev ua raws cai thiab kev kho mob. Cov lus qhia meej txog lub sijhawm tswj hwm kev sib raug zoo nrog cov zaub mov tuaj yeem pab ua kom pom tau cov txiaj ntsig ntau ntawm cov tshuaj.
Ntev -} kev npaj ua tau zoo npaj
Rau ntev - Term cov tswv yim thiab zuam cov khoom siv khoom noj yuav pab tau kev npaj sib nrug thiab ua kom muaj kev tiv thaiv. Qhov no yog qhov tshwj xeeb tshaj yog muab qhov txuas ntxiv ntawm kev ua ntawm Floralaner ntsiav tshuaj.
Tag
Qhov cuam tshuam ntawm cov zaub movNtsiav tshuaj FluralanerKev nqus tau yog qhov tseem ceeb xav hauv cov tshuaj kho tsiaj. Qhov ua tau zoo dua cov kab mob ua ntej thaum tswj cov zaub mov fluralaner, tshwj xeeb} cov rog nyob hauv cov dev mub thiab zuam tiv thaiv. Los ntawm kev nkag siab cov teebmeem khoom noj khoom haus no, cov tswv tsiaj tuaj yeem ua kom zoo dua kev kho mob parasitic tswj thiab cov txiaj ntsig zoo dua rau tsiaj.
Raws li kev tshawb fawb hauv thaj chaw no txuas ntxiv hloov zuj zus, nws yog qhov tseem ceeb kom nyob rau kev paub txog qhov kev pom zoo tshaj plaws thiab kev pom zoo txog kev tswj hwm Fluralaner. Lub ONGPlay ntawm cov zaub mov thiab tshuaj uas tsis kam lees qhov kev nyuaj ntawm cov chaw ua tshuaj nyob rau hauv kev xav txog kev noj zaub mov kom zoo nkauj hauv cov kws kho tsiaj.
Cov FAQ
1. Lub peev xwm tuaj yeem muab cov ntsiav tshuaj Floraner raug muab rau ntawm lub plab khoob?
Thaum cov ntsiav tshuaj fluralaner tuaj yeem muab rau ntawm lub plab khoob, kev tshawb fawb tau qhia tias cov thawj coj noj mov, tshwj xeeb yog cov khoom noj muaj roj thiab cov roj ntsha. Rau kev ua tau zoo tshaj plaws, nws feem ntau pom zoo kom muab cov ntsiav tshuaj nrog lossis tom qab noj mov.
2. Puas yog cov khoom noj cuam tshuam rau kev nqus cov khaub thuas?
Yog lawm, hom khoom noj tuaj yeem cuam tshuam cov kev nqus cov khaub ncaws huv. High - Cov zaub mov muaj roj yuav ua kom tau nqus ntau dua- cov zaub mov muaj roj. Qhov no yog vim lipophilic xwm ntawm fluralaner thiab lub cev hloov pauv uas tsim los ntawm kev noj zaub mov rog.
3. Ntev npaum li cas tom qab noj mov kuv yuav tsum muab kuv tus tsiaj cov ntsiav tshuaj fluralaner?
Rau qhov siab tshaj plaws nqus, nws yog qhov zoo tshaj plaws los tswj hwm tus ntsiav tshuaj Fluralaner thaum lossis tam sim ntawd tom qab noj mov. Txawm li cas los xij, muab cov ntsiav tshuaj hauv 30 feeb ntawm kev pub mis yuav tsum tseem muab cov kev nqus kom haum piv rau kev tswj hwm ntawm lub plab khoob.
Muaj kev paub txog Bloom Tech kom zoo dua: Koj txoj kev tsim txiaj ntawm Fluralaner Ntsiav Tshuaj
Qhov cuam tshuam ntawm cov zaub mov noj ntawm kev nqus ntawm cov ntsiav tshuaj fluralaner yog ib yam uas peb ntawm Bloom Tech zoo siab. Consistently high-quality fluralaner tablets that meet or exceed industry requirements are assured by our state-of-the-art production procedures. Peb txoj kev mob siab rau muab cov khoom uas txhim kho qhov ua tau zoo thiab tus nqi kho tsiaj yog vim kaum xyoo kev tshaj lij hauv kev txawj ntse hauv cov tshuaj saftleutical.
Tsis txhob cia suboptesimal nqus kev nqus koj cov neeg mob tus dev mub thiab zuam tiv thaiv. Xaiv Bloom Tech raws li koj cov chaw tsim khoom Fluralaner Ntsiav Tshuaj. Peb pab neeg kws tshaj lij tau npaj txhij los txhawb koj nrog kev daws teeb meem thiab kev sib twNtses Ntsiav Cov Khaub Ncaws HnavCov. Tiv tauj peb rau hnub noSales@bloomtechz.comXav paub ntau ntxiv txog peb cov khoom lag luam thiab peb yuav ua li cas txhim kho koj li kev saib xyuas tsiaj.
Ntawv Sawv cev
1. Walther, FM, allan, mj, roepke, rk, & nuernberger, mc (2014). Kev Nyab Xeeb ntawm Floranemer chewable ntsiav tshuaj (Bravecto), yog tshiab cov tshuaj tua yeeb yaj kiab, hauv cov dev tom qab tswj hwm qhov ncauj. Parasites & Vectors, 7 (1), 87.
2. Kilp, S., Ramirez, D., Allan, MJ, ROEPKE, RK, & NUNERBERGER, MC (2014). Pharmaconinetics ntawm Fluralaner hauv cov dev tom qab ib qho kev tswj hwm ntawm qhov ncauj lossis lub luag haujlwm. Parasites & Vectors, 7 (1), 85.
3. Taenzler, J., Wengenmayer, C., Williams, J., Zsephiesche, E. ROEPKE, RK, & Heckeroth, thiab Qhov pib ntawm kev ua si ntawm fluralaner (Bravecto ™) tawm tsam centocephaalides ntawm dev. Parasites & Vectors, 7 (1), 567.
4. Gaiens, D., C., Schmidt, M., Hamann, M., J. (2019). Bred - qhov sib txawv hauv cov tshuaj paphaoninetics ntawm Fluralaner hauv cov dev. Phau Ntawv Xov Xwm ntawm Cov Veterinary Medical Media thiab kho, 42 (3), 266-274.

