Shaanxi BLOOM Tech Co., Ltd. yog ib qho ntawm cov tuam ntxhab thiab cov muag khoom ntawm mexidol hmoov hauv Suav teb. Txais tos rau cov lag luam wholesale bulk zoo mexidol hmoov rau muag ntawm no los ntawm peb lub hoobkas. Kev pabcuam zoo thiab tus nqi tsim nyog muaj.
Mexidol, tshuaj hu ua emoxypine succinate (CAS 127464-43-1), yog ib qho hluavtaws derivative ntawm pyridoxine (vitamin B6) uas tau txais kev saib xyuas tseem ceeb hauv kev tshawb fawb kho mob thiab kws tshuaj. Tsim nyob rau hauv Russia, qhov sib xyaw no tau lees paub rau nws cov teebmeem kev kho mob ntau yam, suav nrog cov tshuaj tiv thaiv antioxidant, tiv thaiv ischemic, antihypoxic, thiab cov khoom membranotropic. Mexidol feem ntau yog ua lag luam nyob rau hauv hmoov daim ntawv, pab nws siv nyob rau hauv ntau yam formulations rau qhov ncauj, intravenous, thiab intramuscular tswj.
| Khoom npe | Mexidol hmoov | Mexidol ntsiav tshuaj | Mexidol txhaj | |
| Yam khoom | Hmoov | Tablet | Txhaj tshuaj | |
| Khoom Purity | >98% | >98% | >98% | |
| Khoom Specifications | 1 g yog '; 10 g yog '; 100 g yog '; 1kg ua | Customizable | Customizable | |
| Daim ntawv khoom | Organic synthesis | Customizable | Customizable | |
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| Certificate of Analysis | ||
| Compound npe | Mexidol | |
| CAS Nr. | 127464-43-1 | |
| Ntau | 25kg ua | |
| Chaw tsim tshuaj paus | Shaanxi BLOOM TECH Co., Ltd | |
| Ntau No. | 20250726012 | |
| MFG | Peb Hlis 26, 2025 | |
| EXP | Peb Hlis 26, 2028 | |
| Qauv |
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| Yam khoom | Enterprise txheem | Kev txheeb xyuas qhov tshwm sim |
| Qhov tshwm sim | Dawb rau tawm -dawb | Ua raws |
| Cov ntsiab lus dej | Tsawg dua lossis sib npaug li 5.0% | 0.15% |
| Hnyav Hlau | Pb Tsawg dua lossis sib npaug li 0.5ppm | N.D. |
| Tsawg dua lossis sib npaug li 0.5ppm | N.D. | |
| Hg Tsawg dua lossis sib npaug li 0.5ppm | N.D. | |
| Cd Tsawg dua lossis sib npaug li 0.5ppm | N.D. | |
| Purity (HPLC) | >98% | 99.15% |
| Ib leeg impurity | <0.8% | 0.13% |
| Tag nrho microbial suav | Tsawg dua lossis sib npaug li 750cfu / g | 20 |
| E. Coli | Tsawg dua lossis sib npaug li 2MPN / g | N.D. |
| Salmonella | N.D. | N.D. |
| Ethanol (los ntawm GC) | Tsawg dua lossis sib npaug li 5000ppm | 300 ppm |
| Cia | -80 degree, 2 xyoos; -20 degree, 1 xyoo (Kev kaw cia, deb ntawm noo noo) | |
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| Shaanxi Chuzhan yog lub tuam txhab thev naus laus zis tshwj xeeb hauv kev tshawb fawb thiab kev tsim kho, tsim cov tshuaj thiab cov khoom siv kho kom haum, muab OEM / ODM tag nrho - cov kev daws teeb meem. Peb muab cov kev hloov pauv hloov pauv tag nrho - txheej txheem cov kev pabcuam customized, los ntawm cov qauv kev tshawb fawb thiab kev tsim kho mus rau kev xaiv cov khoom siv, txhua tus tuaj yeem hloov kho raws li cov neeg siv khoom xav tau. Txhawb nqa tag nrho- kev sib koom ua ke ntawm kev sib koom ua ke los ntawm me me- kev sim ntsuas me me, nruab nrab- ntsuas kev sim mus rau loj- nplai ntau lawm, nruab nrog pab pawg kws tshaj lij los muab cov txheej txheem kev ua kom zoo tshaj plaws, thiab tuaj yeem kho cov ntawv ntim raws li cov khoom xav tau ntawm cov neeg siv khoom. | ||
Chemical thiab Physical Properties
Molecular Structure thiab CompositionMexidol yog succinate ntsev ntawm emoxypine, pyridine derivative nrog cov mis molecular C₁₂H₁₇NO₅ thiab molecular hnyav ntawm 255.27 g / mol. Cov qauv muaj 2-ethyl-6-methyl-3-hydroxypyridine moiety txuas rau succinic acid ntawm ester daim ntawv cog lus. Qhov no conjugation txhim khu lub compound stability thiab bioavailability piv rau nws dawb puag daim ntawv. |
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Cov yam ntxwv ntawm lub cevMexidol hmoov zoo nkaus li dawb mus tawm -dawb crystalline khoom nrog lub melting point ntawm kwv yees li 113℃thiab lub boiling point ntawm 280.6℃ntawm 760 mmHg. Nws yog me ntsis soluble hauv dej tab sis dissolves yooj yim hauv cov kuab tshuaj organic xws li ethanol thiab dimethyl sulfoxide (DMSO). Qhov sib xyaw ua ke nthuav tawm qhov tsis muaj zog, nrog lub siab ntawm 0.0022 mmHg ntawm 25 degree, ua rau nws ruaj khov nyob rau hauv cov txheej txheem cia. |
Cia thiab ruaj khovTxhawm rau kom muaj kev ruaj ntseg zoo, Mexidol hmoov yuav tsum tau muab cia rau hauv lub thawv ntim ntawm -20 degree, qhov twg nws khaws cov potency mus txog peb xyoos. Ntawm 4 degree, lub txee lub neej txo qis rau ob xyoos, thaum cov kev daws teeb meem npaj hauv cov kuab tshuaj xws li DMSO lossis saline yuav tsum tau khaws cia ntawm -80℃rau kev siv mus ntev (txog rau lub hlis) lossis -20℃rau kev siv sijhawm luv (ib hlis). Kev raug dej noo thiab lub teeb yuav tsum tau txo kom tsawg kom tsis txhob degradation. |
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Kev siv tshuaj kho mob
Mexidol's versatility tau ua rau nws siv ntau hom kev kho mob, txhawb nqa los ntawm kev sim tshuaj thiab tiag - pov thawj hauv ntiaj teb:
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► Cov Kab Mob Neurological
1) Ischemic Stroke
Mexidol yog dav siv nyob rau hauv mob thiab rov qab theem ntawm ischemic stroke. Ib qho randomized, ob npaug - qhov muag tsis pom, placebo- tswj kev tshawb fawb nrog 120 tus neeg mob tau pom tias Mexidol tau txhim kho cov txiaj ntsig ntawm lub paj hlwb thiab txo qis kev xiam oob qhab thaum noj hauv 24 teev ntawm kev mob stroke. Nws cov tshuaj tiv thaiv -ischemic thiab neuroprotective cuam tshuam tau raug ntaus nqi los txo oxidative kev nyuaj siab thiab txhim kho cov ntshav cerebral.
2) Kev puas tsuaj rau lub hlwb (TBI)
Hauv cov neeg mob TBI, Mexidol ua kom lub hlwb rov zoo thiab txo qhov mob. Kev sim nrog 80 tus neeg mob tau pom tias muaj kev txhim kho tseem ceeb hauv kev nco thiab cov qhab nia siab tom qab 14 hnub ntawm kev kho mob, piv rau cov placebo.
3) Kev paub tsis meej thiab Dementia
Mexidol tau pom cov lus cog tseg hauv kev tswj lub hnub nyoog- cuam tshuam txog kev paub txog kev poob qis thiab vascular dementia. Ib txoj kev tshawb fawb 6- hli hauv cov neeg laus laus uas muaj kev puas siab puas ntsws me me qhia txog kev txhim kho kev nco thiab kev ua haujlwm, yuav yog vim kev txhim kho hippocampal neuroplasticity thiab txo amyloid-beta tsub zuj zuj.
► Psychiatric Disorders
1) Kev ntxhov siab thiab kev nyuaj siab
Mexidol's anxiolytic thiab antidepressant teebmeem tau tshawb pom hauv cov neeg mob uas muaj kev puas siab puas ntsws. Hauv kev sim 56-hnub suav nrog 65 tus neeg mob, Mexidol normalized pw tsaug zog, txhim kho lub siab, thiab txhim kho kev txawj ntse thaum siv nrog kev kho tus qauv. Tshwj xeeb, 40% ntawm cov neeg mob tau pom tias muaj kev txhim kho hauv cov tsos mob ntawm kev ntxhov siab, tsis muaj kev phiv loj heev.
2) Caw Caw Caw Caw Syndrome
Mexidol alleviates tshem tawm cov tsos mob los ntawm modulating GABAergic kis tau tus mob thiab txo oxidative kev nyuaj siab. Ib txoj kev tshawb fawb hauv 45 cawv- cov neeg mob nyob ntawm qhov pom tau tias Mexidol txo qis kev tshee, ntxhov siab, thiab pw tsaug zog zoo dua li diazepam, nrog cov tshuaj sedative tsawg dua.
► Kab Mob plawv
1) Ischemic Heart Disease
Mexidol's anti-ischemic thiab antiarrhythmic zog ua rau nws muaj txiaj ntsig zoo hauv kev tswj hwm angina thiab myocardial infarction. Hauv kev sim nrog 100 tus neeg mob uas tsis ruaj tsis khov angina, Mexidol txo qhov zaus ntawm kev tawm tsam anginal los ntawm 45% thiab txhim kho kev ua haujlwm siab, piv rau trimetazidine, lub npe hu ua metabolic modulator.
2) Peripheral Artery Disease
Mexidol txhim kho cov ntshav khiav mus rau ischemic libs los ntawm kev txhim kho microcirculation thiab txo platelet aggregation. Ib txoj kev tshawb fawb hauv cov neeg mob uas muaj qhov tseem ceeb ntawm cov ceg tawv ischemia tau tshaj tawm cov qhab nia ntawm qhov mob thiab taug kev deb tom qab 3 lub hlis ntawm kev kho mob.
► Ophthalmology
Glaucoma
Mexidol cov teebmeem neuroprotective txuas mus rau cov paj hlwb, ua rau nws muaj peev xwm ntxiv rau hauv kev kho mob glaucoma. Cov kev tshawb fawb tsiaj pom tau hais tias Mexidol txo qis cov kab mob qog nqaij hlav retinal ganglion cell tuag thiab khaws cia qhov muag tsis pom kev, yuav yog los ntawm inhibiting glutamate excitotoxicity thiab oxidative kev nyuaj siab.
Pharmacological Innovations
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► Nanotechnology-Driven Delivery Systems
Mexidol ib nrab luv luv -lub neej (2–2.6 teev) yuav tsum tau noj ntau zaus, txwv tsis pub tus neeg mob ua raws. Yuav kom kov yeej qhov no, cov kws tshawb fawb tab tom tsim cov tshuab nanocarrier. Kev tshawb fawb 2024 encapsulated Mexidol hauv poly (lactic-co-glycolic acid) (PLGA) nanoparticles, ua tiav 3-fold nce hauv hlwb bioavailability thiab tso tawm ntev dua 72 teev hauv cov qauv nas. Ib yam li ntawd, liposomal formulations tau pom cov lus cog tseg hauv kev txhim kho myocardial penetration, nrog rau 2023 mus sib hais qhia txog 40% kev txhim kho hauv ejection feem hauv cov neeg mob plawv tsis ua hauj lwm thaum Mexidol-loaded liposomes tau muab los ntawm kev txhaj tshuaj intracoronary.
► Kev Sib Txuas Kev Kho Mob: Synergistic Approaches
Mexidol lub peev xwm los ua kom muaj zog rau lwm yam tshuaj 'kev cuam tshuam yog tsav kev tshawb fawb kev sib xyaw ua ke. Piv txwv li:
Nrog Citicoline: Hauv post- mob stroke rov qab, Mexidol + citicoline txo qis kev xiam oob qhab los ntawm 22% piv rau kev kho mob monotherapy, yuav yog vim Mexidol's antioxidant teebmeem ntxiv rau citicoline's membrane kho mechanisms.
Nrog Antidepressants: A 2023 meta- kev tshuaj xyuas ntawm 1,200 tus neeg mob pom tias Mexidol augmentation txo kev kho mob- tiv thaiv kev nyuaj siab lub sij hawm los ntawm 35%, ntaus nqi los ntawm nws cov kev hloov pauv ntawm GABAergic thiab serotonergic txoj hauv kev.
Nrog Ozone Therapy: Hauv kev kho mob kub hnyiab, kev sib xyaw ua ke txo kev tuag los ntawm 18% los ntawm ib txhij hais txog oxidative kev nyuaj siab thiab kev kis kab mob, raws li ozone cov tshuaj tua kab mob ntxiv rau Mexidol cov tshuaj tiv thaiv - mob.
► Cov Tshuaj Kho Tus Kheej: Pharmacogenomic Insights
Genetic polymorphisms nyob rau hauv cytochrome P450 enzymes (piv txwv li, CYP2C19) cuam tshuam Mexidol cov metabolism, nrog cov metabolizers tsis zoo uas nthuav tawm 2-fold ntau dua plasma concentrations. Kev sim tshuaj pharmacogenomic tuaj yeem ua kom muaj txiaj ntsig zoo, tshwj xeeb tshaj yog nyob rau hauv cov neeg laus cov neeg mob uas muaj kev phiv xws li kiv taub hau. Tsis tas li ntawd, biomarkers xws li malondialdehyde (MDA) thiab superoxide dismutase (SOD) qib tuaj yeem kwv yees cov lus teb kho mob, tso cai rau cov txheej txheem kev kho mob stratified.
Cov Kev Kho Mob
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► Mexidol nyob rau hauv Acute Ischemic Stroke
1) Keeb Kwm: Mob stroke ischemic yog qhov ua rau tuag thiab kev tsis taus thoob ntiaj teb. Kev cuam tshuam ntxov yog qhov tseem ceeb los txo qis kev puas hlwb hauv hlwb thiab txhim kho cov txiaj ntsig rov qab. Mexidol, nrog nws cov muaj zog antioxidant thiab neuroprotective zog, tau pom cov lus cog tseg hauv cov ntsiab lus no.
2) Kev Kho Mob Scenario: Ib tug 65-xyoo- txiv neej muaj hnub nyoog tshwm sim tshwm sim ntawm sab xis tsis muaj zog thiab hais lus slurred. Ib qho xwm txheej CT scan tau lees paub qhov mob stroke ischemic nyob rau sab laug nruab nrab cerebral hlab ntsha thaj chaw. Tus neeg mob tau muab Mexidol intravenously ntawm ib koob ntawm 250 mg txhua 8 teev, pib li ntawm 6 teev ntawm cov tsos mob tshwm sim, raws li ib feem ntawm cov txheej txheem tswj kev mob stroke.
3) Cov txiaj ntsig: Tom qab 14 hnub ntawm kev kho Mexidol, tus neeg mob tau pom tias muaj kev txhim kho tseem ceeb hauv lub cev muaj zog thiab kev hais lus. Ua raws li- nce MRI scans qhia tau tias txo qhov mob me me thiab txhim kho cerebral perfusion. Tus neeg mob raug tso tawm nrog qhov seem tshuav tsawg kawg nkaus thiab txuas ntxiv Mexidol qhov ncauj (250 mg peb zaug ib hnub) rau 6 lub lis piam ntxiv raws li ib feem ntawm kev kho mob. Cov ntaub ntawv no qhia txog Mexidol lub peev xwm los txhim kho kev rov zoo thiab txo qhov kev tsis taus ntev ntev hauv cov neeg mob ischemic stroke thaum noj ntxov.
► Mexidol in Chronic Cerebrovascular Disease
1) Keeb kwm: Cov kab mob cerebrovascular feem ntau tshwm sim raws li kev paub tsis meej, kev nco tsis zoo, thiab kev puas siab puas ntsws. Mexidol lub peev xwm los txhim kho cerebral metabolism thiab ntshav khiav, nrog rau nws cov tshuaj tiv thaiv antioxidant thiab neuroprotective, ua rau nws yog ib tus neeg sib tw tsim nyog los tswj cov tsos mob no.
2) Kev Kho Mob Scenario: Ib tug poj niam 58-xyoo-laus uas muaj keeb kwm ntawm kev kub siab thiab kev tawm tsam ischemic ib ntus tau nthuav tawm nrog kev nco ploj thiab lub siab hloov pauv xyoo dhau los. Nws tau kuaj pom tias muaj kab mob cerebrovascular ntev nrog kev paub tsis meej. Mexidol tau muab tshuaj ntawm ib koob ntawm 125 mg peb zaug ib hnub ntawm qhov ncauj, nrog rau cov kev kho mob ntshav siab.
3) Cov txiaj ntsig: Tom qab 3 lub hlis ntawm kev kho Mexidol, tus neeg mob tau qhia txog kev nco, kev xav, thiab kev xav zoo. Kev ntsuam xyuas neuropsychological tau lees paub tias muaj kev txhim kho tseem ceeb hauv kev paub txog kev ua haujlwm. Tus neeg mob txuas ntxiv kho Mexidol, thiab nws tus mob tseem nyob ruaj khov nyob rau xyoo tom ntej, tsis muaj kev paub ntxiv lawm. Cov ntaub ntawv no qhia txog Mexidol lub luag haujlwm hauv kev ruaj khov thiab muaj peev xwm txhim kho kev txawj ntse hauv cov neeg mob uas muaj kab mob cerebrovascular.
Mexidol hmoov, los yog emoxypine succinate, yog ib tug hluavtaws derivative ntawm pyridoxine nrog ntau yam tshuaj los. Nws cov antioxidant, antihypoxic, membranotropic, thiab receptor-modulating zog ua rau nws muaj txiaj ntsig zoo rau kev kho mob ntawm ntau yam mob, los ntawm cov kab mob neurological mus rau cov kab mob plawv. Txawm hais tias xav tau kev tshawb fawb ntxiv kom paub meej nws cov txheej txheem ntawm kev nqis tes ua thiab kev siv tshuaj kho mob, kev tshawb fawb thaum ntxov qhia tias Mexidol tuav cov lus cog tseg raws li kev xaiv kev kho mob zoo thiab muaj txiaj ntsig. Raws li lub zej zog kev tshawb fawb txuas ntxiv tshawb fawb txog qhov muaj peev xwm ntawm Mexidol hmoov, nws zoo li cov ntawv thov tshiab thiab tshiab yuav tshwm sim, txuas ntxiv nthuav nws lub luag haujlwm hauv cov tshuaj niaj hnub.
FAQ
1. Mexidol cuam tshuam rau lub hlwb li cas?
Xaus: Cov txiaj ntsig tau qhia tias Mexidol tsis yog tsuas yog muaj kev tiv thaiv ntawm cov neurons, tab sis kuj tuaj yeem txhawb nqa neuroregeneration los ntawm kev nce qib ntawm cov txheej txheem tseem ceeb ntawm cov molecules.
2. Puas yog Maxidol muaj kev nyab xeeb noj txhua hnub?
Noj cov tshuaj no nrog ib khob dej puv nkaus. Nws tuaj yeem noj nrog zaub mov lossis ntawm lub plab khoob. Tsis txhob noj ntau dua 2 ntsiav tshuaj lossis ntsiav tshuaj hauv 24 teev. Naproxen sodium tsuas yog siv rau lub sijhawm luv luv - txog li 5 hnub rau qhov mob thiab 3 hnub ua npaws.
3. Puas yog Mexidol yog cov tshuaj antioxidant?
Cov tshuaj tiv thaiv kab mob ncaj qha ntawm mexidol tau piav qhia, uas suav nrog lub peev xwm ntawm cov tshuaj kom tsis txhob muaj cov dawb radicals thiab ua kom cov haujlwm ntawm cov enzymes antioxidant glutathione peroxidase thiab superoxide dismutase hauv vitro.
Cim npe nrov: Mexidol hmoov, lwm tus neeg, manufacturers, hoobkas, lag luam wholesale, yuav, nqe, tej, kev muag khoom






















